标签归档：抑胃

抑胃酶氨酸-BOC CAS 58521-49-6-AAT Bioquest荧光染料

发表于由

上海金畔生物科技有限公司代理AAT Bioquest荧光染料全线产品，欢迎访问AAT Bioquest荧光染料官网了解更多信息。
抑胃酶氨酸-BOC CAS 58521-49-6价格 7092
产品规格

1 g

产品货号

抑胃酶氨酸-BOC CAS 58521-49-6

产品参数
Ex (nm) – Em (nm) –
分子量 275.34 溶剂 DMF
存储条件 在零下15度以下保存
产品概述

产品基本信息

产品名称：抑胃酶氨酸-BOC

CAS：58521-49-6

储存条件：-15℃避光防潮

保质期：12个月

 

产品物理化学光谱特性

分子量：275.34

溶剂：DMF

激发波长（nm）：N/A

发射波长（nm）：N/A

 

产品介绍

（3S，4S）-Statine是胃蛋白酶抑制剂的新型氨基酸，胃蛋白酶抑制剂是酸性蛋白酶的低分子量抑制剂。这种BOC-Statine构建锁是使用标准BOC化学制备用于药物应用的蛋白酶抗性肽的非常有用的前体。金畔生物是AAT Bioquest的中国代理商，为您提供优质的赖氨酸Lys 5-FITC标记。 

 

参考文献

Investigation of the synthetic route to pepstatin analogues by SPPS using O-protected and O-unprotected statine as building blocks
Authors: Cadicamo CD, Asante V, Abu Ammar M, Borelli C, Korting HC, Koksch B.
Journal: J Pept Sci (2009): 272

[Drug (statine)-induced hepatitis]
Authors: Lazebnik LB, Zvenigorodskaia LA, Khomeriki SG, Efremov LI, Cherkashova EA.
Journal: Eksp Klin Gastroenterol (2009): 110

A simple microscale method for determining the relative stereochemistry of statine units
Authors: Preciado A, Williams PG.
Journal: J Org Chem (2008): 9228

Atovaquone-statine “double-drugs” with high antiplasmodial activity
Authors: Romeo S, Parapini S, Dell’Agli M, Vaiana N, Magrone P, Galli G, Sparatore A, Taramelli D, Bosisio E.
Journal: ChemMedChem (2008): 418

Design, synthesis and SAR of potent statine-based BACE-1 inhibitors: exploration of P1 phenoxy and benzyloxy residues
Authors: Back M, Nyhlen J, Kvarnstrom I, Appelgren S, Borkakoti N, Jansson K, Lindberg J, Nystrom S, Hallberg A, Rosenquist S, Samuelsson B.
Journal: Bioorg Med Chem (2008): 9471

Macrocyclic statine-based inhibitors of BACE-1
Authors: Barazza A, Gotz M, Cadamuro SA, Goettig P, Willem M, Steuber H, Kohler T, Jestel A, Reinemer P, Renner C, Bode W, Moroder L.
Journal: Chembiochem (2007): 2078

Stereocontrolled synthesis of 2,4-diamino-3-hydroxyacids starting from diketopiperazines: a new route for the preparation of statine analogues
Authors: Farran D, Toupet L, Martinez J, Dewynter G.
Journal: Org Lett (2007): 4833

A novel approach to identifying beta-secretase inhibitors: bis-statine peptide mimetics discovered using structure and spot synthesis
Authors: Bridges KG, Chopra R, Lin L, Svenson K, Tam A, Jin G, Cowling R, Lovering F, Akopian TN, DiBlasio-Smith E, Annis-Freeman B, Marvell TH, LaVallie ER, Zollner RS, Bard J, Somers WS, Stahl ML, Kriz RW.
Journal: Peptides (2006): 1877

Molecular docking and 3D-QSAR studies on the binding mechanism of statine-based peptidomimetics with beta-secretase
Authors: Zuo Z, Luo X, Zhu W, Shen J, Shen X, Jiang H, Chen K.
Journal: Bioorg Med Chem (2005): 2121

Design and synthesis of potent inhibitors of the malaria aspartyl proteases plasmepsin I and II. Use of solid-phase synthesis to explore novel statine motifs
Authors: Johansson PO, Chen Y, Belfrage AK, Blackman MJ, Kvarnstrom I, Jansson K, Vrang L, Hamelink E, Hallberg A, Rosenquist A, Samuelsson B.
Journal: J Med Chem (2004): 3353

抑胃酶氨酸-FMOC CAS 158257-40-0-AAT Bioquest荧光染料

发表于由

上海金畔生物科技有限公司代理AAT Bioquest荧光染料全线产品，欢迎访问AAT Bioquest荧光染料官网了解更多信息。
抑胃酶氨酸-FMOC CAS 158257-40-0价格 7092
产品规格

1 g

产品货号

抑胃酶氨酸-FMOC CAS 158257-40-0

产品参数
Ex (nm) – Em (nm) –
分子量 397.47 溶剂 DMF
存储条件 在零下15度以下保存
产品概述

产品基本信息

产品名称：抑胃酶氨酸-FMOC

CAS：158257-40-0

储存条件：-15℃避光防潮

保质期：12个月

 

产品物理化学光谱特性

分子量：397.47

溶剂：DMF

激发波长（nm）：N/A

发射波长（nm）：N/A

 

产品介绍

(3S,4S)-Statine是新发现的抑肽素（胃蛋白酶抑制剂）上的氨基酸，一种小分子量酸性蛋白酶抑制剂。在制药的过程中使用FMOC化学标准，FMOC-Statine是制备抑制蛋白酶的多肽的非常有用的前体。金畔生物是AAT Bioquest的中国代理商，为您提供优质的赖氨酸Lys 5-FITC标记。 

 

参考文献

Investigation of the synthetic route to pepstatin analogues by SPPS using O-protected and O-unprotected statine as building blocks
Authors: Cadicamo CD, Asante V, Abu Ammar M, Borelli C, Korting HC, Koksch B.
Journal: J Pept Sci (2009): 272

[Drug (statine)-induced hepatitis]
Authors: Lazebnik LB, Zvenigorodskaia LA, Khomeriki SG, Efremov LI, Cherkashova EA.
Journal: Eksp Klin Gastroenterol (2009): 110

A simple microscale method for determining the relative stereochemistry of statine units
Authors: Preciado A, Williams PG.
Journal: J Org Chem (2008): 9228

Atovaquone-statine “double-drugs” with high antiplasmodial activity
Authors: Romeo S, Parapini S, Dell’Agli M, Vaiana N, Magrone P, Galli G, Sparatore A, Taramelli D, Bosisio E.
Journal: ChemMedChem (2008): 418

Design, synthesis and SAR of potent statine-based BACE-1 inhibitors: exploration of P1 phenoxy and benzyloxy residues
Authors: Back M, Nyhlen J, Kvarnstrom I, Appelgren S, Borkakoti N, Jansson K, Lindberg J, Nystrom S, Hallberg A, Rosenquist S, Samuelsson B.
Journal: Bioorg Med Chem (2008): 9471

Macrocyclic statine-based inhibitors of BACE-1
Authors: Barazza A, Gotz M, Cadamuro SA, Goettig P, Willem M, Steuber H, Kohler T, Jestel A, Reinemer P, Renner C, Bode W, Moroder L.
Journal: Chembiochem (2007): 2078

Stereocontrolled synthesis of 2,4-diamino-3-hydroxyacids starting from diketopiperazines: a new route for the preparation of statine analogues
Authors: Farran D, Toupet L, Martinez J, Dewynter G.
Journal: Org Lett (2007): 4833

A novel approach to identifying beta-secretase inhibitors: bis-statine peptide mimetics discovered using structure and spot synthesis
Authors: Bridges KG, Chopra R, Lin L, Svenson K, Tam A, Jin G, Cowling R, Lovering F, Akopian TN, DiBlasio-Smith E, Annis-Freeman B, Marvell TH, LaVallie ER, Zollner RS, Bard J, Somers WS, Stahl ML, Kriz RW.
Journal: Peptides (2006): 1877

Molecular docking and 3D-QSAR studies on the binding mechanism of statine-based peptidomimetics with beta-secretase
Authors: Zuo Z, Luo X, Zhu W, Shen J, Shen X, Jiang H, Chen K.
Journal: Bioorg Med Chem (2005): 2121

Design and synthesis of potent inhibitors of the malaria aspartyl proteases plasmepsin I and II. Use of solid-phase synthesis to explore novel statine motifs
Authors: Johansson PO, Chen Y, Belfrage AK, Blackman MJ, Kvarnstrom I, Jansson K, Vrang L, Hamelink E, Hallberg A, Rosenquist A, Samuelsson B.
Journal: J Med Chem (2004): 3353

抑胃酶氨酸STATINE CAS 49642-07-1-AAT Bioquest荧光染料

发表于由

上海金畔生物科技有限公司代理AAT Bioquest荧光染料全线产品，欢迎访问AAT Bioquest荧光染料官网了解更多信息。
抑胃酶氨酸STATINE CAS 49642-07-1价格 2823
产品规格

100 mg

产品货号

抑胃酶氨酸STATINE CAS 49642-07-1

产品参数
Ex (nm) – Em (nm) –
分子量 175.23 溶剂 DMF
存储条件 在零下15度以下保存
产品概述

产品基本信息

产品名称：抑胃酶氨酸STATINE

CAS：49642-07-1

储存条件：-15℃避光防潮

保质期：12个月

 

产品物理化学光谱特性

分子量：175.23

溶剂：DMF

激发波长（nm）：N/A

发射波长（nm）：N/A

 

产品介绍

抑胃酶氨酸是一种新发现的抑肽素（胃蛋白酶抑制剂）上的氨基酸，一种小分子量酸性蛋白酶抑制剂。金畔生物是AAT Bioquest的中国代理商，为您提供优质的赖氨酸Lys 5-FITC标记。 

 

参考文献

Investigation of the synthetic route to pepstatin analogues by SPPS using O-protected and O-unprotected statine as building blocks
Authors: Cadicamo CD, Asante V, Abu Ammar M, Borelli C, Korting HC, Koksch B.
Journal: J Pept Sci (2009): 272

[Drug (statine)-induced hepatitis]
Authors: Lazebnik LB, Zvenigorodskaia LA, Khomeriki SG, Efremov LI, Cherkashova EA.
Journal: Eksp Klin Gastroenterol (2009): 110

A simple microscale method for determining the relative stereochemistry of statine units
Authors: Preciado A, Williams PG.
Journal: J Org Chem (2008): 9228

Atovaquone-statine “double-drugs” with high antiplasmodial activity
Authors: Romeo S, Parapini S, Dell’Agli M, Vaiana N, Magrone P, Galli G, Sparatore A, Taramelli D, Bosisio E.
Journal: ChemMedChem (2008): 418

Design, synthesis and SAR of potent statine-based BACE-1 inhibitors: exploration of P1 phenoxy and benzyloxy residues
Authors: Back M, Nyhlen J, Kvarnstrom I, Appelgren S, Borkakoti N, Jansson K, Lindberg J, Nystrom S, Hallberg A, Rosenquist S, Samuelsson B.
Journal: Bioorg Med Chem (2008): 9471

Macrocyclic statine-based inhibitors of BACE-1
Authors: Barazza A, Gotz M, Cadamuro SA, Goettig P, Willem M, Steuber H, Kohler T, Jestel A, Reinemer P, Renner C, Bode W, Moroder L.
Journal: Chembiochem (2007): 2078

Stereocontrolled synthesis of 2,4-diamino-3-hydroxyacids starting from diketopiperazines: a new route for the preparation of statine analogues
Authors: Farran D, Toupet L, Martinez J, Dewynter G.
Journal: Org Lett (2007): 4833

A novel approach to identifying beta-secretase inhibitors: bis-statine peptide mimetics discovered using structure and spot synthesis
Authors: Bridges KG, Chopra R, Lin L, Svenson K, Tam A, Jin G, Cowling R, Lovering F, Akopian TN, DiBlasio-Smith E, Annis-Freeman B, Marvell TH, LaVallie ER, Zollner RS, Bard J, Somers WS, Stahl ML, Kriz RW.
Journal: Peptides (2006): 1877

Molecular docking and 3D-QSAR studies on the binding mechanism of statine-based peptidomimetics with beta-secretase
Authors: Zuo Z, Luo X, Zhu W, Shen J, Shen X, Jiang H, Chen K.
Journal: Bioorg Med Chem (2005): 2121

Design and synthesis of potent inhibitors of the malaria aspartyl proteases plasmepsin I and II. Use of solid-phase synthesis to explore novel statine motifs
Authors: Johansson PO, Chen Y, Belfrage AK, Blackman MJ, Kvarnstrom I, Jansson K, Vrang L, Hamelink E, Hallberg A, Rosenquist A, Samuelsson B.
Journal: J Med Chem (2004): 3353